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Table 5 Drug-likeness properties of compounds 1–10 by the SwissADME server

From: Drug repurposing of pyrazolotriazine derivatives as potential anti-SARS-CoV-2 agents: in vitro and in silico studies

Compound

Lipinski

Ghose

Veber

Egan

Muegge

Bioavailability

score

1

Yes

Yes

Yes

Yes

Yes

0.55

2

Yes

Yes

Yes

Yes

Yes

0.55

3

Yes

Yes

Yes

Yes

Yes

0.55

4

Yes

Yes

Yes

Yes

Yes

0.55

5

Yes

Yes

Yes

Yes

Yes

0.55

6

Yes

Yes

Yes

Yes

Yes

0.55

7

Yes

Yes

Yes

Yes

Yes

0.55

8

Yes

Yes

Yes

Yes

Yes

0.55

9

Yes

No

Yes

Yes

No

0.55

10

Yes

No

Yes

Yes

No

0.55